2025

Genetic deletion of the purinergic receptor P2rx7 worsens the phenotype of α‑sarcoglycan muscular dystrophy.
Astigiano, Cecilia, Principi, Elisa, Pintus, Sara, Benzi, Andrea, Baratto, Serena, Panicucci, Chiara, Passalacqua, Mario, Sierra-Marquez, Juan, Nicke, Annette ORCID: https://orcid.org/0000-0001-6798-505X, Antonini, Francesca, Del Zotto, Genny, Cicatiello, Annunziata Gaetana, Raffaghello, Lizzia, Rezzonico Jost, Tanja, Grassi, Fabio, Bruzzone, Santina ORCID: https://orcid.org/0000-0003-2034-3716, Bruno, Claudio and Gazzerro, Elisabetta ORCID: https://orcid.org/0000-0003-2428-0302
ACS Pharmacology & Translational Science 8 (10): 3477-3489. 10 October 2025

Selectivity and safety characterization of a xanthine-imidazothiazole lead structure: a novel tryptophan hydroxylase inhibitor of peripheral serotonin synthesis.
Wesolowski, R. ORCID: https://orcid.org/0009-0002-7228-1051, Schütz, A. ORCID: https://orcid.org/0000-0002-0606-2574, Lisurek, M. ORCID: https://orcid.org/0009-0004-7685-5387, Nazaré, M. ORCID: https://orcid.org/0000-0002-1602-2330, Heinemann, U. ORCID: https://orcid.org/0000-0002-8191-3850, Pleimes, D., Bader, M. ORCID: https://orcid.org/0000-0003-4780-4164 and Specker, E. ORCID: https://orcid.org/0000-0002-9471-9520
ACS Pharmacology & Translational Science 8 (6): 1678-1693. 13 June 2025

2021

Viewpoints on the first transatlantic GPCR symposium for early-career investigators.
Bender, B.J., Bock, A. ORCID: https://orcid.org/0000-0002-6344-6494, Nesheva, D.N. and Perry-Hauser, N.A.
ACS Pharmacology & Translational Science 4 (5): 1705-1711. 8 October 2021

2020

Ligand-specific allosteric coupling controls G-protein-coupled receptor signaling.
Holze, J., Bermudez, M. ORCID: https://orcid.org/0000-0002-7421-3282, Pfeil, E.M., Kauk, M., Bödefeld, T., Irmen, M., Matera, C. ORCID: https://orcid.org/0000-0001-6939-3859, Dallanoce, C. ORCID: https://orcid.org/0000-0002-7383-1484, De Amici, M., Holzgrabe, U. ORCID: https://orcid.org/0000-0002-0364-7278, König, G.M. ORCID: https://orcid.org/0000-0003-0003-4916, Tränkle, C., Wolber, G. ORCID: https://orcid.org/0000-0002-5344-0048, Schrage, R., Mohr, K., Hoffmann, C., Kostenis, E. ORCID: https://orcid.org/0000-0001-8284-5514 and Bock, A. ORCID: https://orcid.org/0000-0002-6344-6494
ACS Pharmacology & Translational Science 3 (5): 859-867. 9 October 2020

The European Research Network on Signal Transduction (ERNEST): toward a multidimensional holistic understanding of G protein-coupled receptor signaling.
Sommer, M.E. ORCID: https://orcid.org/0000-0003-0493-8584, Selent, J. ORCID: https://orcid.org/0000-0002-1844-4449, Carlsson, J. ORCID: https://orcid.org/0000-0003-4623-2977, De Graaf, C. ORCID: https://orcid.org/0000-0002-1226-2150, Gloriam, D.E., Keseru, G.M., Kosloff, M., Mordalski, S., Rizk, A., Rosenkilde, M.M. ORCID: https://orcid.org/0000-0001-9600-3254, Sotelo, E. ORCID: https://orcid.org/0000-0001-5571-2812, Tiemann, J.K.S. ORCID: https://orcid.org/0000-0001-7551-6245, Tobin, A. ORCID: https://orcid.org/0000-0002-1807-3123, Vardjan, N., Waldhoer, M. and Kolb, P. ORCID: https://orcid.org/0000-0003-4089-614X
ACS Pharmacology & Translational Science 3 (2): 361-370. 10 April 2020